Momwe mungagwiritsire ntchito mankhwala a Aspirin Cardio?

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Aspirin Cardio amagwiritsidwa ntchito pofuna kupewa thrombosis, kugunda kwa mtima, komanso kubwezeretsa thupi pambuyo pakuchita opaleshoni yamtima kapena mitsempha yamagazi. Mapiritsi amathandizira kubwezeretsa magazi mu ubongo.

Ath

Anatomical-achire-mankhwala gulu (ATX) - B01AC06.

Mu Latin, dzina la mankhwalawa limamveka motere - Aspirin Cardio.

Aspirin Cardio amagwiritsidwa ntchito pofuna kupewa thrombosis, kugunda kwa mtima, komanso kubwezeretsa thupi pambuyo pakuchita opaleshoni yamtima kapena mitsempha yamagazi.

Kutulutsa mafomu ndi kapangidwe kake

Aspirin C ndi piritsi yoyera yozungulira yomwe ili enteric. Mankhwalawa amapezeka mu kuchuluka kwa 100 kapena 300 mg. Katoniyo amakhala ndi matuza awiri kapena anayi, kutengera kuchuluka kwa mapiritsi (10 kapena 14).

Zomwe zili piritsi zimaphatikizidwa ndi zomwe zimagwira - acetylsalicylic acid. 1 pc akaunti ya 300 kapena 100 mg ya chinthucho. Opezekapo ndi monga:

  • cellulose ufa - 10 kapena 30 mg;
  • wowuma chimanga - 10 kapena 30 mg.

Zomwe chipolopolocho chimakhala ndi:

  • kopolymer wa methaconic acid ndi ethacrylate 1: 1 (Eudragit L30D) - 7.857 kapena 27, 709 mg; polysorbate 80 - 0,186 kapena 0,514 mg;
  • sodium lauryl sulfate - 0,057 kapena 0,157 mg;
  • talc - 8.1 kapena 22.38 mg;
  • triethyl citrate - 0,8 kapena 2.24 mg.

Zotsatira za pharmacological

Mankhwalawa amatanthauza ma pinkillers ndi anti-yotupa mankhwala (non-steroidal) ndi mankhwala omwe amakhudza minofu metabolism (antiplatelet agent).

Pharmacological kanthu - anti-kophatikiza. Zomwe zimachitika Aspirin Cardio zimagwirizanitsidwa ndi mphamvu ya thupi yogwira. Chifukwa chotseka ma cell a prostaglandinsynthetase, ma enzyme omwe amaphatikizidwa ndi prostaglandin biosynthesis, kupanga mahomoni opatsirana kumalepheretsa. Chifukwa chake, mankhwalawa amatha kukhala ndi zotsatira za analgesic, antipyretic komanso anti-yotupa.

Aspirin Cardio amagwiritsidwa ntchito pofuna kupewa thrombosis, kugunda kwa mtima, komanso kubwezeretsa thupi pambuyo pakuchita opaleshoni yamtima kapena mitsempha yamagazi.

Kupezeka kwa thrombosis kumachepetsedwa chifukwa chakuti chinthu chogwira ntchito chimachepetsa kutsatira zomatira komanso zomatira zamapulatifomu. Aspirin amakhudza kuthekera kwa madzi am'magazi ku fibrinolysis komanso amachepetsa kuchuluka kwa zomwe zikuchitika. Imabwezeretsa ntchito yam'magazi.

Mukamamwa mankhwalawa, chiwopsezo cha maselo amitsempha ku zinthu zomwe zimakwiyitsa zimachepa.

Izi zikuchitika chifukwa cha kuchepa kwa chiwerengero cha otetezereka omwe amakhala onyamula kukwiya. Kutha kupanga antipyretic kwenikweni.

Pharmacokinetics

Pambuyo acetylsalicylic acid amalowa m'thupi, chinthucho chimatengedwa m'mimba. Pa mayamwidwe, chigawo chogwira chimadutsa mu metabolite - salicylic acid. Thupi limapukusidwa mu chiwindi ndi ma enzymes monga phenyl salicylate, glucuronide salicylate ndi salicyluric acid, omwe amapezeka minofu yambiri komanso mkodzo.

Chifukwa chochepa chochita ndi mayendedwe am'madzi mu seramu ya akazi, njira ya metabolic imachepetsedwa. ASA imatheka mu plasma ya mphindi 10-20 mutatha kugwiritsa ntchito, salicylic acid - pambuyo 30-60 Mphindi.

ASA imatetezedwa ndi chipolopolo chosagwira asidi, kotero mankhwalawa samatulutsidwa m'mimba, koma m'malo amchere wa duodenum. Mafuta a Acid amachepetsa pofika maola 3-6, mosiyana ndi mapiritsi opanda othandizira.

Ma acid amamangidwa ndi mapuloteni a plasma ndipo amafalikira thupi lonse. Salicylic acid imatha kulowa mkati mwa placenta ndikuchotseredwa mkaka wa m'mawere. Thupi limachotsedwa m'thupi pakhungu. Ndi kachitidwe koyenera ka thupi, mankhwalawa amachotsedwa pakatha masiku 1-2 ndikugwiritsa ntchito kamodzi.

Ndi kachitidwe koyenera ka thupi, mankhwalawa amachotsedwa pakatha masiku 1-2 ndikugwiritsa ntchito kamodzi.

Zomwe zimathandiza

Mankhwala ndi mankhwala otsatirawa:

  1. Njira zodzitchinjiriza kwa pachimake myocardial infaration pamaso pangozi. Izi ndi monga: matenda a shuga, matenda oopsa, kunenepa kwambiri (kunenepa kwambiri), ukalamba, kumwa pafupipafupi zinthu za nikotini.
  2. Angina pectoris, kuphatikizapo mitundu yokhazikika komanso yosakhazikika.
  3. Hypovolemia.
  4. Vuto la mtima.
  5. Matenda oopsa.
  6. Kuteteza kwa Stroko
  7. Matenda a hememologic.
  8. Kuwonongeka kwa kufalikira kwa ubongo, ischemic kuwonongeka kwa ubongo.
  9. Chiwopsezo cha kugunda kwam'mimba kwambiri ndi ma pulmonary embolism, kuphatikizapo nthambi zake.
  10. Kupewa kwa thromboembolism pambuyo pa opaleshoni yamatumbo.

Mankhwalawa amathandizidwanso chifukwa cha ngozi za cerebrovascular, kuwonongeka kwa ubongo wa ischemic.

Contraindication

Kugwiritsa ntchito mankhwalawa osavomerezeka mu milandu iyi:

  • Hypersensitivity zigawo zikuluzikulu za mankhwala;
  • mphumu
  • kuphwanya kwam'mimba khunyu (zilonda zam'mimba, magazi am'mimba);
  • zaka za ana;
  • nthawi yoyamwitsa;
  • mimba
  • hepatic, aimpso ndi mtima kulephera.

Ndi chisamaliro

Mukamamwa pamodzi ndi mankhwala angapo, musanachite opaleshoni (mankhwalawa angayambitse kuchepa kwa magazi), munthawi yachitatu ya mimba.

Chenjezo limayenera kumwa mapiritsi musanachitike opaleshoni (mankhwalawa angayambitse kuchepa kwa magazi).

Momwe angatenge

Tengani mankhwalawo monga adalimbikitsira ndi dokotala kapena mogwirizana ndi malangizo. Amayikidwa mkati, osambitsidwa ndi madzi ambiri. Ngati angafune, piritsiyo imaphwanyidwa ndikusungunuka m'madzi. Ngakhale ndikulimbikitsidwa kuti mumwe mankhwalawo osaperera, kwathunthu.

Nthawi yanji

Mapiritsi amalimbikitsidwa musanadye.

Kutalika bwanji

Njira ya chithandizo imayikidwa ndi dokotala. Pogwiritsa ntchito nthawi yayitali, kuledzera kwa thupi kumatha kuchitika.

Ndi matenda ashuga

Kudya tsiku lililonse mankhwala tikulimbikitsidwa.

Zotsatira zoyipa

Mlingo wowerengeka molakwika wa mankhwala ungayambitse zotsatira zoyipa kuchokera mthupi lonse.

Mlingo wowerengeka molakwika wa mankhwala ungayambitse zotsatira zoyipa kuchokera mthupi lonse.

Matumbo

Kusanza, kupweteka pamtima, kusanza, kudula ululu pamimba. Nthawi zambiri, zotupa m'mimba.

Hematopoietic ziwalo

Kuchulukitsa kwa magazi munthawi ya ntchito, mapangidwe a zilonda, magazi kuchokera pamphuno, kwamkodzo thirakiti, magazi m'mimba. Pali umboni wamatumbo am'mimba, magazi am'mimba.

Pakati mantha dongosolo

Chizungulire, kupweteka mutu, tinnitus, kumva kwakanthawi kwamakutu.

Kuchokera kwamikodzo

Matenda a impso, osowa kwambiri aimpso.

Matupi omaliza

Zochitika pakhungu (zotupa, kuyabwa, matenda a Addison), kutupa kwa mphuno, chifuwa, kusokonezeka kwa dongosolo la kupuma (mphumu, kusokonezeka kwa anaphylactic).

Mlingo wowerengeka molakwika wa mankhwalawa ungayambitse kudwala kwam'mimba.
Ngati bongo, kufalikira kwa mphuno.
Mlingo wolakwika wa mankhwalawa umayambitsa mutu.
Ngati bongo, aimpso kukanika kumachitika, kawirikawiri - aimpso kulephera.
Kugwiritsa ntchito molakwika mankhwalawa kumayambitsa khungu (zotupa, kuyabwa, matenda a Addison).

Malangizo apadera

Mankhwalawa ayenera kugwiritsidwa ntchito motsogozedwa ndi dokotala. Zotsatira zoyipa ndi mankhwala osokoneza bongo ndizowopsa kwa okalamba.

Kuyenderana ndi mowa

Acid ndi zakumwa zoledzeretsa sizigwirizana. Kugwiritsa ntchito munthawi yomweyo kumatha kuyambitsa mavuto (kumawonjezera kukakamiza, kukulitsa matenda amtima), kumachepetsa kuchiritsa kwamankhwala.

Zokhudza mphamvu pakuwongolera njira

Zisakhudze kuthekera koyendetsa magalimoto.

Gwiritsani ntchito panthawi yoyembekezera komanso mkaka wa m`mawere

Mankhwalawa amakhudza kwambiri njira ya kubereka komanso kukula kwa mwana wosabadwayo.

Kutenga mankhwala osokoneza bongo oposa 300 mg / tsiku mu 1 trimester ya mimba kumayambitsa kusintha kwa pathologies mu fetus. Mu 3 trimester, kumwa mapiritsi kungayambitse kuletsa kwabwino, kuchulukitsa kwa magazi mwa mayi ndi mwana wosabadwayo. Mwana amatha kudwala matenda a m'matumbo ndipo amwalira nthawi yomweyo ngati mankhwalawo aledzera asanaperekedwe. Chifukwa chake, kumwa mankhwalawa panthawiyi ndikotsutsana.

Mankhwalawa amakhudza kwambiri njira ya kubereka komanso kukula kwa mwana wosabadwayo.

Mu trimester yachiwiri, wodwalayo amatha kutenga Aspirin atatha kuwunika chiopsezo ku thanzi la mayi ndi mwana wosabadwayo ndi katswiri. Mlingo sayenera kupitirira 150 mg / tsiku.

Ndi kumwa kwa kanthawi kochepa kwa mankhwalawa, kuyamwitsa sikungayimitsidwe, chifukwa kuchuluka kochepa kwa zinthu zamankhwala kumalowa mkaka, zomwe sizimayambitsa zovuta m'mwana. Pogwiritsa ntchito mapiritsi nthawi yayitali mukamayamwa, kudyetsa kuyenera kuyimitsidwa mpaka zinthu zitachotsedwa mthupi la mayi.

Kupangira Aspirin Cardio kwa Ana

Mankhwala osavomerezeka kuti agwiritsidwe ntchito ndi ana ochepera zaka 15 omwe ali ndi matenda opumira kwambiri oyambitsidwa ndi matenda. Izi zimaphatikizidwa ndi chiopsezo cha Reye syndrome.

Popanda matenda, dokotalayo amakupatsani mankhwala malinga ndi kuchuluka kwa thupi la mwanayo komanso matenda ake. Mankhwala ogwiritsa ntchito kamodzi amagwiritsidwa ntchito.

Kulimbitsa mtima wamtima, tikulimbikitsidwa kumwa Taurine.

Mankhwala osavomerezeka kuti agwiritsidwe ntchito ndi ana ochepera zaka 15 omwe ali ndi matenda opumira kwambiri oyambitsidwa ndi matenda.

Gwiritsani ntchito mu ukalamba

Kulandila kuyenera kuchitika malinga ndi malingaliro a dokotala pakakhala kuti pali contraindication. Nthawi zambiri ntchito kukalamba kupewa matenda a mtima.

Bongo

Ndi poyizoni wofatsa kapena wapakati, zizindikiro zotsatirazi zimawonekera:

  • Chizungulire
  • thukuta;
  • kusanza, kusanza
  • chisokonezo.

Ngati zizindikiro zikapezeka, pitani kuchipatala. Asanapereke chithandizo chamankhwala, kugwiritsa ntchito kaboni yokhazikitsidwa mobwerezabwereza, kubwezeretsa kuchuluka kwa madzi kumalimbikitsidwa.

Ngati zizindikiro zikapezeka, pitani kuchipatala. Asanapereke chithandizo chamankhwala, kugwiritsa ntchito kaboni yokhazikitsidwa mobwerezabwereza, kubwezeretsa kuchuluka kwa madzi kumalimbikitsidwa.

Woopsa milandu bongo:

  • kuchuluka kwa kutentha kwa thupi;
  • kulephera kupuma;
  • kuphwanya mtima, impso, chiwindi;
  • tinnitus, ugonthi;
  • Kutaya magazi kwa GI.

Kuchiza kumafuna wodwala kuchipatala.

Kuchita ndi mankhwala ena

Pogwiritsa ntchito munthawi yomweyo, zochita za mankhwala otsatirawa zimakulitsidwa:

  1. Methotrexate.
  2. Heparin ndi anticoagulants osadziwika.
  3. Digoxin.
  4. Othandizira a Hypoglycemic.
  5. Valproic acid.
  6. NSAIDs.
  7. Ethanol (kuphatikizapo zakumwa zoledzeretsa).

Pogwiritsa ntchito munthawi yomweyo, zotsatira za Methotrexate zimatheka.

Amachepetsa mphamvu ya mankhwalawa zotsatirazi:

  1. Zodzikongoletsera.
  2. ACE zoletsa.
  3. Ndi uricosuric zotsatira.

Analogi

Zotsatira za mankhwalawa zimaphatikizapo: Cardiask, Upsarin UPSA, Thrombo ACC, Cardiomagnyl. Ngati ndi kotheka, Aspirin amayenera kugwiritsidwa ntchito ngati adokotala adafotokoza.

Kukhala wamkulu! Zinsinsi zotengera mtima wa mtima. (12/07/2015)
Aspirin: maubwino ndi zopweteketsa | Dr. Butchers
Okwatirana omwe afa. Cardiac Aspirin ndi NSAIDs. Kukhala wamkulu! (11/18/2015)

Kodi pali kusiyana kotani pakati pa Aspirin ndi Aspirin Cardio

  • zikuchokera mankhwala;
  • wokutira Aspirin Cardio ndi nembanemba wapadera kuteteza nembanemba wam'mimba thirakiti kuti lisawonongeke;
  • Mlingo
  • mtengo.

Kupita kwina mankhwala

Popanda mankhwala a dokotala.

Mtengo wa Aspirin Cardio

Ku Russia, mtengo wamankhwala umasiyanasiyana 90 mpaka 276 rubles.

Kusunga mankhwala Aspirin Cardio

Sungani ku kutentha kosaposa 25 ° C.

Tsiku lotha ntchito

Zaka 5

Ndemanga pa Aspirin Cardio

Valera, wazaka 49, Volgograd: "Dotolo amamuwonetsa mankhwala ochepetsa magazi pakakhala vuto la magazi. Zinthu zakhala zikuyenda bwino, koma nthawi zina zimadzetsa kutentha."

Svetlana, wazaka 33, Mozhaysk: "Pamodzi ndi zotsatira zabwino, zotsatira zoyipa zikuwonekeranso. Sindinathe kumwa mankhwala: kupweteka kwam'mimba, chizungulire chanthawi zambiri zinayamba.

Oleg, wazaka 44, Norilsk: "Anapatsidwa mapiritsi a zovuta zamitsempha yamiyendo. Ndinachotsa matendawa. Palibe zotsatira zoyipa."

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