Latren ndi gulu la zotumphukira vasodilators. Amagwiritsidwa ntchito muzochita zamankhwala kuti akwaniritse vasodilating. Njira yothandizirana motere ndiyofunikira kubwezeretsa magazi moyenera m'malo omwe akukhudzidwa ndi minofu ndikuthandizira magazi. Mankhwala amathandiza kuthetsa thrombosis, atherosulinosis ndi zovuta za choroid wa ocular organ.
Dzinalo Losayenerana
Pentoxifylline.
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Latren amathandizira kuthetsa thrombosis, atherosclerosis ndi zovuta za choroid wa ocular organ.
ATX
C04AD03.
Kutulutsa mafomu ndi kapangidwe kake
Mankhwala amapangidwa mu mawonekedwe a yankho pokonzekera kulowetsedwa. Fomu ya mulingo uli m'malo opezeka magalasi okhala ndi 100, 200 kapena 400 ml ya yogwira - pentoxifylline. Mowoneka, yankho lake ndi madzi owoneka bwino a chikasu pang'ono kapena wopanda utoto. Zowonjezera zina zowonjezera kusintha kwa mayamwidwe, mawonekedwe amadzimadzi a sodium lactate, madzi osalala a jakisoni, potaziyamu ndi sodium chloride, calcium chloride amagwiritsidwa ntchito.
Zotsatira za pharmacological
Pentoxifylline imapangidwa kuchokera ku methylxanthine; ndi ya gulu la zotumphukira vasodilators. Pharmacological zimachitika chifukwa chopinga cha phosphodiesterase. Mofananamo, mankhwala amtunduwu amathandizira kuti pakhale 3,5-AMP mu minofu yosalala ya mtima endothelium, ma cell am'magazi, zimakhala ndi ziwalo.
Pentoxifylline imalepheretsa kudziphatika kwa maselo ofiira am'magazi ndi ma cell am'magazi, imapatsa mphamvu komanso imawonjezera kukana kwa maselo awo. Chifukwa cha kuchepa kwa kuphatikiza, mawonekedwe amwazi amachepa, mphamvu ya fibrinolytic imawonjezeka ndipo zofunikira za magazi zimasintha.
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Recre Latrena amathandizira kuti matenda a mtima asinthe.
Pentoxifylline imathandizira kuwonjezeka kwa plasma ndende ya fibrinogen. Pankhaniyi, chinthu chogwira chimachepetsa kukana konsekonse m'matumbo a zotumphukira, zimakhala ndi mphamvu yofowoka yam'mitsempha. Kumwa mankhwalawa kumathandizira kusintha kwamtima. Chifukwa chokwaniritsa njira yochizira, kuchuluka kwa magazi m'magawo a ischemic kumawonjezera: mwayi wokhala ndi vuto la kuchepa kwa oxygen m'maselo amachepa, minofu imalandira mpweya wokwanira ndi michere.
Mu maphunziro azachipatala, kuchuluka kwa mankhwalawa pa kama wodwala m'magawo a m'mphepete, dongosolo lamanjenje, komanso kuchuluka kwa mitsempha yolembedwa. Mankhwalawa ali ndi mphamvu yofooka pakukula kwa ziwiya zama coronary.
Pharmacokinetics
Pamene pentoxifylline ilowa m'mitsempha yamagazi, imafika m'magazi okwanira 60 maminiti. Pakadutsa koyamba kudzera mu hepatocytes, chinthu chogwira ntchito chimasinthika kwathunthu. Zinthu zowola zimaposa kuchuluka kwambiri kwa plasma ya pentoxifylline nthawi 2 ndipo zimakhala ndi achire. Hafu ya moyo ndi maola 1.6. 90% ya mankhwalawa amachoka m'thupi mwa ma metabolites, 4% imachotsedwera ndowe m'njira yake yoyamba.
Zizindikiro zogwiritsidwa ntchito
Pentoxifylline ndi vasodilator yomwe imasintha ntchito yogwira ntchito ya capillaries. Mankhwalawa amathandizira kumasula minofu ya minyewa yosalala yamitsempha yamagazi, bronchospasm. Vasodilator amalembedwa kuti azingokhala ndi vuto la m'maganizo kumbuyo kwa kusintha kwa kusintha kwa mtima kwa endothelium. Mankhwalawa amathandizira kuwonjezera magazi mu gawo la zilonda zam'mimba kapena malo okhala m'munsi.
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Mankhwala amathandiza pa matenda a occlusive matenda a zotumphukira mitsempha ya matenda ashuga ndi atherosulinotic etiology:
- kuphwanya trophic minofu;
- kupweteka m'misempha ya miyendo ndikupuma;
- kudalirana pang'ono;
- mitsempha ya varicose.
Mankhwalawa amabwezeretsanso kufalikira kwa magazi ndi ziwalo zamagazi kumkhutu, zimathandizira kuthetsa thrombosis ndikuwongolera minyewa yamitsempha motsutsana ndi matenda a shuga a polyneuropathy. Mankhwalawa amagwiritsidwa ntchito pochiza matenda a Raynaud.
Contraindication
Mankhwalawa amaletsedwa kuperekedwa kwa anthu omwe ali ndi hypersensitivity ku zinthu zomwe zimapanga maziko a Latren, ndi xanthine. Mankhwala ali osavomerezeka ntchito pamaso matenda ndi zotsatirazi matenda:
- magazi akulu;
- hemorrhagic diathesis;
- makonzedwe achitukuko kapena kukhalapo kwa pachimake myocardial infarction;
- matenda a porphyrin;
- hemorrhege
- pathological mtima mungoli zosokoneza;
- kusintha kwakukulu kwa atherosclerotic mu endothelium yam'mimba ndi mitsempha ya m'magazi;
- kuthamanga kwa magazi;
- matenda am'mimba.
Mankhwala ali osavomerezeka kwa anthu omwe ali ndi chiwindi komanso impso.
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Ndi chisamaliro
Anthu odwala ulcerative-erosive zotupa m'mimba ndi duodenum ayenera kuyan'ana mkhalidwe wamatenda a mankhwalawa panthawi ya mankhwala ndi Latren. Chenjezo limaperekedwa kwa anthu omwe ali ndi vuto la mtima komanso pamaso pa matenda a shuga. Mankhwalawa amawayang'aniridwa poyang'aniridwa mosamalitsa pambuyo pakuchita opaleshoni yambiri.
Momwe mungatenge Latren
Mankhwalawa amaperekedwa kudzera m'mitsempha monga kulowetsedwa. Mlingo wakhazikitsidwa ndi dokotala wokhudzana ndi njira ya pathological ndi mawonekedwe a wodwala. Zotsatirazi ndi monga kulemera kwa thupi, zaka, matenda opatsirana, kulolerana kwa mankhwala, kuopsa kwa zovuta zamagazi.
Odwala opitirira zaka 12 akulimbikitsidwa kuyika dontho ndi 100-200 ml ya mankhwalawa. Kuyendetsa madontho kumapitilizidwa kwa maola 1.5-3. Ndi kulekerera kwabwino, kuchuluka kwa mlingo mpaka 400-500 ml (wofanana ndi 300 mg) wa jekeseni ndikuloledwa.
Mlingo woyenera wololedwa tsiku lililonse ukufika 500 ml. Nthawi zambiri, mankhwalawa amatha masiku pafupifupi 5-7. Ngati ndi kotheka, kupitiliza chithandizo kumasinthidwa kukamwa kwa vasodilators pamapiritsi.
Ndi matenda ashuga
Mankhwala amatha kupititsa patsogolo mphamvu ya hypoglycemic ya mankhwala antidiabetes, chifukwa chake, munthawi ya mankhwalawa ndi Latren, ndikofunikira kuyendetsa kuchuluka kwa shuga m'magazi ndikunyamula shuga. Zotsirizazo ndikofunikira kuti muchepetse kukula kwa hypoglycemia.
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Zotsatira zoyipa Latrena
Zotsatira zoyipa zimachitika ndi mlingo woyenera wa mankhwalawa.
Pa mbali ya gawo la masomphenyawo
Mwina kuchepa kwa maonedwe acuity, kutupa kwa conjunctiva, zotupa za m'mimba, kutsatiridwa ndi kutulutsa. Nthawi zina, kuwonongeka kwa mawonekedwe kumayendera limodzi ndi kukula kwa scotoma.
Kuchokera minofu ndi mafupa
Nthawi zina, minyewa imayamba kufooka.
Matumbo
Pogaya chakudya chambiri, munthu amayamba kumva kugundana, kusanza. Nthawi zina, kuphwanya matumbo motility, kutupa kwa chiwindi kumayamba, cholecystitis imakulaku. Kuwoneka kwa cholestasis ndikotheka.
Hematopoietic ziwalo
Kuletsa kwamitsempha ya hematopoiesis kumayendera limodzi ndi kuchepa kwa maselo ofiira am'magazi ndi ma cell, komwe kungayambitse kukula kwa hypoplastic anemia. Muzovuta kwambiri, pamakhala chiopsezo cha kufa.
Pakati mantha dongosolo
Ndi mulingo woyipa, mutu umayamba kumva kuti mumva chizungulire, pamutu, kupsinjika, minofu kukokana, kusokonezeka kwa tulo. Munthu amakhala ndi nkhawa zopanda pake.
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Kuchokera ku kupuma
Mwina kukula kwa kufupika kwa mpweya.
Pa khungu
Khungu limakhudzana ndi zotupa, kuyabwa, erythema ndi matenda a Stevens-Johnson. Kusokonekera kwa maula a msomali kumakulitsidwa.
Kuchokera pamtima
Wodwalayo amayamba kumva kutuluka, kutupa kwa miyendo. Pali tachycardia, kusinthasintha kwa magazi. Zikakhala zowopsa, magazi amatha kutuluka.
Kuchokera kumbali ya kagayidwe
Mwina chitukuko cha matenda a anorexia, kuchepa kwa potaziyamu, thukuta ndi kuwonjezeka kwa kutentha kwa thupi, ntchito ya michere ya chiwindi imachulukirachulukira.
Matupi omaliza
Thupi lawo siligwirizana limodzi ndi khungu ndi anaphylactoid zimachitika.
Zokhudza mphamvu pakuwongolera njira
Poona kuchepa kotheka kwa kuthamanga kwa ma psychomotor komanso kuwonongeka kwakanthawi panthawi yamankhwala, ndikofunikira kupewa kuyendetsa galimoto ndi zida zovuta.
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Malangizo apadera
Pankhani ya lupus erythematosus ndi ma pathologies ena ofunikira minofu, ndikofunikira kupereka mankhwala pokhapokha pakuwunikira mozama mapindu ake ndi zoopsa zake. Kuyesedwa kwa magazi pafupipafupi kumafunikira chifukwa choopsa cha kuchepa magazi m'thupi.
Odwala omwe ali ndi vuto la mtima wosalephera amafunika kufikira gawo la kubwezeretsa magazi musanagwiritse ntchito mankhwala.
Odwala omwe akuyembekezeka kukula kwa anaphylactic zimayesedwa kuti ayesere kulolera mankhwala. Pofuna kuchitapo kanthu, mankhwala amasiya.
Gwiritsani ntchito mu ukalamba
Anthu azaka zosaposa 50 ayenera kusamala.
Kulembera Latren kwa ana
Ana osaposa zaka 12 sakonda mankhwala a Latren. Kwa ana, ndikofunikira kuwerengera mulingo molingana ndi kulemera kwa thupi - 10 ml ya mankhwalawa pa 1 makilogalamu a kulemera. Kwa ana akhanda, mlingo wa tsiku ndi tsiku amawerengedwa mofananamo, koma mlingo waukulu sayenera kupitirira 80-100 ml.
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Gwiritsani ntchito pa nthawi yoyembekezera komanso mkaka wa m`mawere
Palibe deta pamatumbo a pentoxifylline komanso momwe zimakhalira pakukula kwa embryonic. Chifukwa chake, kulowetsedwa kwa mtsempha wa mankhwalawa kumayikidwa pokhapokha ngati milandu ya vasodilating ikhoza kulepheretsa moyo wa mayi. The achire zotsatira ayenera kupitilira chiwopsezo cha intrauterine michere mu mluza.
Pa yoyamwitsa, poika Latren, ndikofunikira kusiya kuyamwa.
The ntchito aimpso kuwonongeka
Matenda a impso amalimbikitsa theka la moyo wa mankhwalawa, chifukwa chake, kulowetsedwa kwa Latren kumaloledwa kokha pamaso pa matenda a impso komanso olimbitsa.
Gwiritsani ntchito ntchito yolakwika ya chiwindi
Mankhwalawa saloledwa kugwiritsidwa ntchito ndi anthu omwe akuwonongeka kwambiri kwa chiwindi.
Latren Zambiri
Ndi mankhwala osokoneza bongo, zizindikiro zotsatirazi zimayamba:
- kufooka kwa minofu;
- Chizungulire
- minyewa yamanjenje;
- dontho la kuthamanga kwa magazi;
- chisokonezo ndi kutayika kwa chikumbumtima;
- kuchuluka kwa mtima;
- kuthira nkhope;
- kusanza ndi mseru;
- magazi ndi kukha magazi kulowa m'matumbo am'mimba;
- minofu kukokana;
- malungo.
Wovutitsidwayo amafunikira kuchipatala mwachangu. Chithandizo chimathandizira kupewa kutulutsa magazi mkati ndi kuthetsa zizindikiro za bongo.
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Kuchita ndi mankhwala ena
Pentoxifylline imatha kubweretsa kuchepa kwa kuchuluka kwa shuga m'magazi pogwiritsa ntchito othandizira a hypoglycemic kapena insulin. Chifukwa chake, odwala matenda a shuga ayenera kufunsana ndi endocrinologist kuti asinthe mlingo wa mankhwala antidiabetes.
Pochita malonda pambuyo pake, pakhala pali kuchepa kwa kugunda kwa magazi ndi kugwiritsidwa ntchito kofanana ndi ma antivitamini K, anticoagulants achindunji komanso osagwirizana ndi Latren. Mukaphatikizidwa ndi mankhwalawa, kuyang'anira ntchito ya anticoagulant ndikofunikira.
Pentoxifylline imathandizira antihypertensive mphamvu ya antihypertensive mankhwala. Zotsatira zake, ochepa hypotension angachitike.
Kusagwirizana kwakuthupi kumawonedwa ndikusakanikirana kwa Latren ndi njira zina zamafuta mu syringe yomweyo.
Chithandizo chogwira ntchito chimachulukitsa mulingo wa Theophylline, ndichifukwa chake kuchulukitsa kapena kuwonjezera kuchuluka kwa mawonekedwe owoneka chifukwa chogwiritsa ntchito Theophylline.
Kuyenderana ndi mowa
Mankhwala sangaphatikizidwe ndi mankhwala omwe amakhala ndi ethanol komanso mankhwala omwe amamwa mowa. Mowa wa Ethyl ndiwotsutsana ndi pentoxifylline, amalimbikitsa kutsata kwa maselo ofiira amwazi, kuletsa magazi. Ethanol imayambitsa vasospasm komanso kukula kwa thrombosis. Pali kusowa achire zotsatira ndi kuwonongeka.
Analogi
Mndandanda wa mankhwala omwe ali ndi mankhwala ofanana kapena mankhwala:
- Trental;
- Bilobil;
- Pentoxifylline;
- Maluwa;
- Agapurin;
- Pentilin.
Kupita kwina mankhwala
Mankhwalawa sagulitsidwa popanda chiwonetsero chachipatala mwachindunji.
Kodi ndingagule popanda kulandira mankhwala?
Chithandizo chamankhwala chimafunikira chifukwa kugulitsa kwaulere kwa Latren ndikochepa. Mlingo wolakwika wa vasodilator ungayambitse bongo kapena zotsatira zoyipa kwambiri.
Mtengo
Mtengo wapakati wa kulowetsedwa umasiyanasiyana 215 mpaka 270 rubles.
Zosungidwa zamankhwala
Ndikofunikira kusunga vutoli pamtunda wa + 2 ... + 25 ° C m'malo owuma, olekanitsidwa ndi dzuwa.
Tsiku lotha ntchito
Zaka 2
Wopanga
Yuri-Farm LLC, Russia.
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Ndemanga
Ulyana Tikhonova, wazaka 56, St. Petersburg
Anapereka yankho la thrombosis. Poyamba, omwe akutsikira a Latren adaphatikizidwa ndi jakisoni wa heparin, pambuyo pake amasinthidwa ndikumwa mapiritsi. Kulowetsedwa kunathandiza kupukusa magazi, kutupa kutapita. Ndikuganiza kuphatikiza mtengo wamtengo ndi mtundu. Panalibe zovuta zilizonse, koma ndinayenera kusiya mowa ndi kusuta munthawi ya chithandizo. Dokotala adati atsatire mosamalitsa malangizo ogwiritsa ntchito kuti achepetse zovuta zaumoyo.
Leopold Kazakov, wazaka 37, Ryazan
Ndinalemba mankhwala a Latren ndi otolaryngologist, kwa omwe ndidadandaula kuti amachepera kumva acuity ndi mawonekedwe a tinnitus wofuula. Cholinga chake chinali kukula kwa dystonia. Ma infusions adathandizira kuthetsa kupweteka kwa mutu, ndikulira m'makutu. Ndazindikira kuti masomphenyawa anali abwinobwino. Zotsatira zoyipa zimawoneka ngati njira yochepetsera kuthamanga kwa magazi. Kuti awathetse, kuchepetsa mlingo wake kunafunikira. Dokotala wopezekapo ayenera kusintha. Sindikukulangizani kuti musinthe nokha paokha, chifukwa pali chiopsezo cha mankhwala osokoneza bongo ambiri.