Mankhwala Methylethylpyridinol: malangizo ntchito

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The pharmacological zimatha mankhwala Methylethylpyridinol amalola ntchito mu neurology, mtima ndi ophthalmology. Mankhwalawa ndi a gulu la angioprotectors, omwe ndi ofunika kwambiri pakukhudzana kwa matenda a mtima ndi mtima.

Dzinalo Losayenerana

Methylethylpyridinol (Methylethylpiridinol).

Pharmacological zimatha mankhwala Methylethylpyridinol amalola ntchito mu neurology.

ATX

C05CX - mankhwala ena omwe amachepetsa kubwereza kwa capillary.

Kutulutsa mafomu ndi kapangidwe kake

Mankhwalawa amapezeka mu mawonekedwe a yankho la makolo. Ndiwisi wopanda mafuta. Chosakaniza chophatikizika ndi methylethylpyridinol hydrochloride. 1 ml ya yankho, 10 mg ya thunthu.

Zinthu zothandiza ndi yankho la hydrochloric acid ndi madzi a jakisoni.

Yankho limagulitsidwa mu ampoules, 5 kapena 10 zidutswa phukusi lililonse.

Mbale zokhala ndi madontho amaso zimapezeka pansi pa mayina ena ogulitsa.

Zotsatira za pharmacological

Mankhwala ali ndi vuto linalake poletsa kusintha kwakanema. Zomwe zimagwiritsidwa ntchito zikuwonetsa izi:

  1. Zoteteza. Vasodilation imachitika, mtundu wa microcirculation umakhala bwino. The permeability wa mtima makoma amakhala munjira, kagayidwe mu minofu yamitsempha yamagazi imayatsidwa, kutupa kwa minofu kumachotsedwa.
  2. Antioxidant. Njira za lipid oxidation ndizoletsa. Mlingo wachitukuko cha kusintha kokhudzana ndi zaka umachepetsedwa, chiopsezo chotenga ma pathologies a khansa.
  3. Antiaggregant. Kuchepa kwa magazi kuwundana kumachepetsedwa. Chithandizo chogwira ntchito chimalepheretsa kuphatikiza mapulateleti, chimathandizira kusungunuka kwa mawonekedwe a fibrin. Ili ndi zotupa m'mimba, imakhazikika pa index ya prothrombin ndi heestasis.
  4. Antihypoxic. Kuthamanga kwa magazi ndi kayendedwe ka oksijeni m'misempha imakhala yofanana. Pazovuta zam'magazi, kuwonongeka kwa mitsempha kumachepa, kukana kwa maselo ku ischemia ndi hypoxia kumawonjezeka.
  5. Kuyambiranso. Amasintha kukoka kwam'mimba ndikusinthanso kwamatumbo m'matumbo amaso. Zowopsa zoyipa kwambiri pa retina zimalephereka.

The pharmacology ya mankhwala ndi chifukwa cha activation wa kagayidwe kachakudya njira kagayidwe. Pali mathamangitsidwe amitundu mitundu, kukondoweza kwa kusinthika kwa minofu.

Mankhwala ali ndi vuto linalake poletsa kusintha kwakanema.

Pharmacokinetics

Mu thupi, chinthu chogwira chimalowa m'matipi onse. Zimapukusidwa mu chiwindi, zotsalira zimatsitsidwa ndi kwamikodzo dongosolo. Ndi mtsempha wamkati, theka la moyo ndi mphindi 18.

Zizindikiro zogwiritsidwa ntchito

Mankhwala ndi mankhwala limodzi. Mankhwalawa amagwiritsidwa ntchito motere:

  1. Mothandizidwa ndi mtima, amadziwitsidwa kupewa matenda obwezeretsanso kumbuyo kwa kubwezeretsa kutuluka kwa magazi, mankhwalawa osakhazikika a angina ndi kupweteka kwapakati pachimake. Mankhwala bwino kugwira ntchito ndi kukomoka kwa mtima, amachepetsa ischemic kuwonongeka kwa mtima minofu. Mankhwalawa amachepetsa zomwe zimachitika mu mtima.
  2. Amagwiritsidwa ntchito mu neurosurgery ndi neurology kwa ischemic ndi hemorrhagic stroke, matenda osakhalitsa komanso ozungulira a matenda amitsempha yamagazi, komanso pochiza kuvulala kwamitsempha. Amagwiritsidwa ntchito pakukonzanso pambuyo pakugwiritsidwa ntchito kwa hematomas opweteka kwambiri komanso ozungulira. Ndi kuthamanga kwa magazi, mankhwalawa amakhala ndi vuto lothetsa magazi, amachepetsa chiopsezo chotaya magazi. Kuphwanya ma dysfunctions kwa autonomic kumakonzedwa, ndipo kubwezeretsa kwa kuphatikiza kwa ubongo kumathandizira.
  3. Mu ophthalmology, amalembera subconjunctival ndi intraocular hemorrhages, hemorrhage mu anterior chipinda cha maso ndi sclera, angioretinopathy, dystrophic keratitis, mawonekedwe owuma a angiosselotic macular degeneration. Mankhwalawa retinal thrombosis, mavuto a myopia ndi myopia, chorioretinal dystrophy, matenda a m'matumbo. Amayikiratu dystrophy, kuvulala ndi kuwotchedwa kwa cornea, mutavala magalasi olumikizana - - kuti muteteze cornea ndi retina kuti asayang'ane ndi kuwala. Mankhwalawa amagwiritsidwa ntchito pambuyo pochita opaleshoni ya glaucoma ndi njira zina zochitira opaleshoni.

Kuchiza ndi mankhwalawa kumachitika moyang'aniridwa ndi adokotala.

Mu cardiology, methylethylpyridinol ndi mankhwala wothandiza kupewa reperfusion.
Mu neurosurgery ndi neurology, mankhwalawa amagwiritsidwa ntchito ngati ischemic stroke.
Mu ophthalmology, methylethylpyridinol amalembera subconjunctival ndi intraocular hemorrhages.

Contraindication

Mankhwalawa adapangidwa kuti azigwiritsidwa ntchito osakwana zaka 18, azimayi oyembekezera komanso oyembekezera. Mankhwalawa sangathe kugwiritsidwa ntchito ngati mukuwona zizindikiro za hypersensitivity.

Ndi chisamaliro

Kugwiritsa ntchito kumafuna kusamala kwapadera pakakhala vuto la magazi, chizolowezi chowonetsa matendawa, pakuchita opaleshoni, pakakhala zizindikiro za magazi kwambiri.

Momwe mungatenge methylethylpyridinol?

Kugwiritsa ntchito mankhwalawa kumaphatikizapo njira zingapo zoyendetsera:

  • mtsempha wamitseko;
  • mu mnofu
  • subconjunctival;
  • chithunzi
  • kubwezera;
  • kukhazikitsa mu gawo la conjunctival.

Kubayira ndi dontho kumachitika ndi akatswiri odziwa ntchito zachipatala. Ndi kukapanda kuleka, mankhwalawa amayamba kusungunulidwa ndi yankho la dextrose kapena sodium chloride.

Kukonzekera kumayendetsedwa ndi malangizo omwe ali ndi malingaliro ambiri ogwiritsira ntchito mankhwalawa. Kutalika kwa maphunziro muzochitika zosiyanasiyana ndiku kuyambira 3 mpaka 30 masiku. Njira zochizira ndi mulingo wothetsera vutoli zimaperekedwa ndi dokotala aliyense payekha.

Ndi kukapanda kuleka, mankhwalawa amayamba kusungunulidwa ndi yankho la dextrose kapena sodium chloride.

Ndi matenda ashuga

Mkufufuza kwa asayansi, zinavumbulutsidwa kuti kugwiritsa ntchito yankho motsutsana ndi mtundu wa matenda a shuga I kumapangitsa kuti ntchito zamapulatini zizigwira bwino, ndizosangalatsa zomwe zidawoneka pokhudzana ndi kusokonekera kwa endothelial. Chifukwa chake, mankhwalawa amagwiritsidwa ntchito mu zovuta za matenda a matenda ashuga nephropathy.

Zotsatira zoyipa za Methylethylpyridinol

Ndi mtsempha wamkati, titha kumverera. Mu ophthalmology, jakisoni ungayambitse conjunctival hyperemia, kutsekeka kwa minofu ya paraorbital zone. Izi zimadutsa palokha.

Poyerekeza ndi chithandizo cha mankhwalawa ndi mankhwalawa, kusapeza bwino m'mimba ndi dera la epigastric ndikotheka, nseru nthawi zina zimadziwika.

Pakati mantha dongosolo

Kukhumudwa kwakanthawi kochepa kumatha kuchitika, ndipo mutu ndi kugona kungachitike.

Kuchokera pamtima

Nthawi zina, pamakhala kuchuluka kwa kuthamanga kwa magazi, kumva kupweteka mumtima.

Matupi omaliza

Zotsatira zoyipa zam'deralo zimadziwika ndi zotupa pakhungu, kuyabwa ndi kuyaka.

Khansa yambewu imawonedwa chifukwa cha mankhwala a Methylethylpyridinol.
Poyerekeza ndi momwe mankhwalawo amathandizira ndi mankhwala, kusapeza bwino m'mimba ndi dera la epigastric ndikotheka.
Kutenga Methylethylpyridinol, mutu umayamba.
Kugona kumawerengedwa ngati mbali imodzi yamankhwala.
Nthawi zina, pamakhala kuchuluka kwa magazi chifukwa chogwiritsa ntchito mankhwalawa Methylethylpyridinol.
Zochita za m'deralo zimakhala ndi zotupa pakhungu.
Zotsatira zoyipa za mankhwalawa, kumva kupweteka m'dera la mtima kumatha kuonekera.

Zokhudza mphamvu pakuwongolera njira

Ndikulimbikitsidwa kusiya ntchito zomwe zimafunikira chisamaliro chambiri komanso kuthamanga kwa mayankho panthawi yayitali ya chithandizo.

Malangizo apadera

Pa chithandizo ndi mankhwalawa, ndikofunikira kuyang'anira kuchuluka kwa magazi ndi kuthamanga kwa magazi.

Gwiritsani ntchito mu ukalamba

Kwa odwala okalamba, mlingo umayang'aniridwa ndi adokotala. Mankhwala nthawi zambiri zotchulidwa ophthalmology kupewa ndi kuchiza matenda a m'matumbo, zotupa mu sclera.

Kupatsa ana

Osaperekedwa kwa anthu osakwana zaka 18.

Gwiritsani ntchito pa nthawi yoyembekezera komanso mkaka wa m`mawere

Kugwiritsa ntchito yankho la azimayi oyembekezera komanso oyamwitsa sikumaperekedwa chifukwa cha kusowa kwa maphunziro pazotsatira za chinthu pa mwana wosabadwayo ndi mwana pa nthawi yokumwitsa. Ngati pakufunika thandizo la mankhwala, mwayi woti mugwiritse ntchito umayesedwa ndi adokotala.

Mankhwala ochulukirapo a Methylethylpyridinol

Kuchulukitsa Mlingo wovomerezeka kumawonjezera zovuta za zotsatira zoyipa. Palibe mankhwala, mankhwalawa amaphatikizapo mankhwala opatsirana, kuphatikizapo kumwa mankhwala omwe ali ndi vuto la hypotensive. Kuyang'anira kuthamanga kwa magazi kumafunika.

Mankhwala sayenera kusakanikirana ndi mankhwala ena.

Kuchita ndi mankhwala ena

Mphamvu ya antioxidant ya mankhwalawa imalimbikitsa mphamvu za vitamini E.

Mankhwala sayenera kusakanikirana ndi mankhwala ena. Palibe mankhwala omwe amagwirizana ndi mankhwala ena.

Kuyenderana ndi mowa

Zakumwa zoledzeretsa zam'kati mwa mankhwala siziyenera kupatula. Mowa umawonjezera mitsempha yamagazi ndipo umalepheretsa mitsempha. Kuyanjana kumeneku kumapangitsa kuti ntchitoyo ikhale yothandiza komanso kumathandizanso kuti mankhwalawo athe kugwira bwino ntchito.

Analogi

Pali mitundu ingapo ya ma analogues, omwe amaphatikizanso zomwezo:

  • Emoxipin (jakisoni ndi madontho amaso);
  • Vixipin (maso akutsikira 5 ml);
  • Emoxy optics (maso akutsikira 5 ml);
  • Emoxibel (diso limatsika 5 ml, jakisoni njira 1% ndi 3%);
  • Emoxipin-Acti (yankho la kulowetsedwa).

Ma Analogs molingana ndi makina ochitira zinthu ndi kukonzekera kochokera pa Ethylmethylhydroxypyridineced (Mexicoidol, Mexico, Neurox, ndi zina).

Mankhwala amatha kukhala ndi mawonekedwe ogwiritsa ntchito. Kuthekera kwa kulowetsa mankhwala kuyenera kukambidwa ndi dokotala.

Emoxipin
Vixipine
Vixipine
Dokotala wamaso
Emoxibel
Mexicoidol
Achimor
Neurox

Kupita kwina mankhwala

Mankhwala ndi a gulu la mankhwala omwe amapezeka.

Kodi ndingagule popanda kulandira mankhwala?

M'mafakisoni, tchuthi ndi mankhwala.

Mtengo wa methyl ethyl pyridinol

Mtengo wapakatikati wa ma CD ndi ma ruble 20-80.

Zosungidwa zamankhwala

Mankhwalawa amayenera kusungidwa m'malo amdima pa kutentha osaposa 25ºC.

Tsiku lotha ntchito

Alumali moyo zaka 3 kuyambira tsiku kupanga.

Wopanga

Mankhwalawa amapangidwa ndi makampani angapo aku Russia, kuphatikiza Eskom, Ozone, Atoll ndi Ellara.

Methylethylpyridinol nthawi zina amatha kusintha m'malo mwa mankhwala Emoxy-optic.
Emoxybel amadziwika ngati analogue ya mankhwala a Methylethylpyridinol.
Emoxipin amadziwika ngati analogue ya mankhwala a Methylethylpyridinol.
Mndandanda wa mankhwala Methylethylpyridinol ndi Vixipin.
Malinga ndi limagwirira ntchito, Neurox amadziwika kuti ndi analog ya methylethylpyridinol.
Mexicoidol imachita chimodzimodzi ndi Methylethylpyridinol.
Mexicor ndi analogue ya mankhwala Methylethylpyridinol.

Ndemanga za Methylethylpyridinol

Petr Valerievich, katswiri wa zamitsempha, ku Moscow: "Muzochita zamankhwala, mankhwalawa amagwiritsidwa ntchito kawirikawiri pazovuta zamagazi. Mankhwala okwera mtengo komanso othandiza."

Marianna Alekseevna, katswiri wa ophthalmologist, Penza: "Njira yothandiza pochiritsira matenda angapo a ophthalmology ndi njira yothetsera jakisoni. Madontho amaso amatha kugwiritsidwa ntchito ndi wodwalayo kunyumba monga momwe adanenera adotolo. Komabe, amagulitsidwa pansi pa dzina lina."

Vitaliy, wazaka 50, Saratov: "Dotolo adapereka mankhwala opangira jakisoni wa matenda amtima. madokotala. "

Julia, wazaka 42, Murmansk: "Dotolo adauza amayi kuti apereke yankho m'maso ndi chorioretinitis. Mwanjira iyi, mankhwalawo amagulitsidwa m'masitolo ogulitsa dzina lina. Ubwino wa mankhwalawa ndiwotsika mtengo, wotsika mtengo."

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